Publications

IL-1β stimulates a novel axis within the NFκB pathway in endothelial cells regulated by IKKα and TAK-1

Craig Rachel, McIntosh Kathryn, Ho Ka Ho, McCulloch Ashley, Riley Christopher, Lawson Christopher, MacKay Simon P, Paul Andrew, Coats Paul, Plevin Robin

Biochemical Pharmacology Vol 232 (2025)

https://doi.org/10.1016/j.bcp.2024.116736

Design and synthesis of novel aminoindazole-pyrrolo[2,3-b]pyridine inhibitors of IKKα that selectively perturb cellular non-canonical NF-κB signalling

Riley Christopher, Ammar Usama, Alsfouk Aisha, Anthony Nahoum G, Baiget Jessica, Berretta Giacomo, Breen David, Huggan Judith, Lawson Christopher, McIntosh Kathryn, Plevin Robin, Suckling Colin J, Young Louise C, Paul Andrew, Mackay Simon P

Molecules Vol 29 (2024)

https://doi.org/10.3390/molecules29153515

Synthesis and evaluation of small molecule inhibitors of the androgen receptor N-terminal domain

Henry Martyn C, Riley Christopher M, Hunter Irene, Elwood Jessica M L, Lopez-Fernandez J Daniel, Minty Laura, Coe Diane M, McEwan Iain J, Jamieson Craig

ACS Medicinal Chemistry Letters Vol 14, pp. 1800-1806 (2023)

https://doi.org/10.1021/acsmedchemlett.3c00426

Current and emerging approaches to noncompetitive AR inhibition

Riley Christopher M, Elwood Jessica M L, Henry Martyn C, Hunter Irene, Lopez-Fernandez J Daniel, McEwan Iain J, Jamieson Craig

Medicinal Research Reviews Vol 43, pp. 1701-1747 (2023)

https://doi.org/10.1002/med.21961

More publications